SCHEMBL4764953

SCHEMBL4764953

[CH2]C[C@H](C)CC(=O)N(CC1=Nc2ccccc2CC1=O)C1CCCNCC1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 19/20 0.38
SLC6A4 P31645 19/20 0.38
SLC6A3 Q01959 11/20 0.38
KCNH2 Q12809 3/20 0.38
CYP2D6 P10635 2/20 0.35
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768429 0.90 SLC6A2 (0.38) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL4830403 0.71 HTR4 (0.35) ALDH1A1
SCHEMBL19358932 0.65 GBA1 (0.45) SLC6A4
SCHEMBL22387506 0.61 SLC6A2 (0.51) SLC6A2SLC6A4SLC6A3KCNH2ALDH1A1
SCHEMBL6595138 0.61 SLC6A4 (0.32) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL27787052 0.59 OPRM1 (0.65) SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL11371357 0.58 ALDH1A1 (0.45) ALDH1A1
SCHEMBL27196422 0.58 CYP4F2 (0.46) ALDH1A1
SCHEMBL27787053 0.57 SLC6A4 (0.61) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL3811903 0.57 DCUN1D1 (0.58) SLC6A2SLC6A4SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed