SCHEMBL4765880

SCHEMBL4765880

NS(=O)(=O)c1cccc(NC2=NC(=O)C(=Cc3cccc4cccnc34)S2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.43
ALOX5 P09917 1/20 0.40
CA9 Q16790 3/20 0.39
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA4 P22748 1/20 0.38
CCNT1 O60563 4/20 0.38
CDK1 P06493 4/20 0.38
CCNB1 P14635 4/20 0.38
CDK9 P50750 4/20 0.38
MAPK1 P28482 1/20 0.38
CCNA2 P20248 4/20 0.37
CDK2 P24941 4/20 0.37
CDK7 P50613 2/20 0.37
CCNH P51946 2/20 0.37
CCNA1 P78396 2/20 0.37
CCNE1 P24864 1/20 0.37
CCND3 P30281 1/20 0.37
FLT3 P36888 1/20 0.37
CDK6 Q00534 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2788506 0.85 CSNK2A2 (0.45) ROCK1ALOX5CA9CA1CA2
SCHEMBL2788502 0.85 CSNK2A2 (0.45) ROCK1ALOX5CA9CA1CA2
SCHEMBL4770645 0.82 NEK2 (0.39) CCNT1CDK9CDK2CCNE1
SCHEMBL4772646 0.79 KMT2A (0.52) CA9CA1CA2CA4KMT2A
SCHEMBL4774422 0.78 CYP2C9 (0.36) MEN1KMT2AL3MBTL1
SCHEMBL4768062 0.74 DYRK3 (0.38) MEN1KMT2AL3MBTL1
SCHEMBL4776074 0.74 NPC1 (0.35) MEN1KMT2AL3MBTL1
SCHEMBL4768194 0.73 BACE1 (0.36) MEN1KMT2AL3MBTL1
SCHEMBL4776063 0.72 NQO1 (0.43) CCNT1CDK9FLT3CDK6SLC2A1
SCHEMBL4770530 0.71 PDE10A (0.46) MAPK1MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567112-B1 THIAZOLIDIN-4-ONES FOR INHIBITING hYAK3 PROTEINS SMITHKLINE BEECHAM CORP (US) 2008-10-15 EP claimed