SCHEMBL4776063

SCHEMBL4776063

CN1CCN(c2ccc(NC3=NC(=O)C(=Cc4cccc5cccnc45)S3)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 2/20 0.43
EGFR P00533 2/20 0.43
TNIK Q9UKE5 2/20 0.42
JAK2 O60674 1/20 0.41
JAK3 P52333 1/20 0.41
DYRK3 O43781 2/20 0.41
CLK1 P49759 2/20 0.41
CLK2 P49760 2/20 0.41
CLK3 P49761 2/20 0.41
GSK3B P49841 2/20 0.41
DYRK1A Q13627 2/20 0.41
DYRK2 Q92630 2/20 0.41
CLK4 Q9HAZ1 2/20 0.41
DYRK1B Q9Y463 2/20 0.41
CSNK1E P49674 1/20 0.41
DYRK4 Q9NR20 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 1/20 0.40
RAB9A P51151 1/20 0.40
CCNT1 O60563 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765576 0.86 CHKA (0.41) TNIKJAK2JAK3CCNT1CDK4
SCHEMBL2787956 0.84 EGFR (0.52) NQO1EGFRTNIKDYRK3CLK1
SCHEMBL2787952 0.84 EGFR (0.52) NQO1EGFRTNIKDYRK3CLK1
SCHEMBL4774422 0.77 CYP2C9 (0.36) L3MBTL1KDM4ERAB9AALDH1A1MAPT
SCHEMBL4765880 0.72 ROCK1 (0.43) JAK3L3MBTL1CCNT1CDK9CDK6
SCHEMBL4770645 0.72 NEK2 (0.39) CCNT1CDK9MAPT
SCHEMBL2788132 0.71 CHKA (0.51) EGFRDYRK3CLK1CLK3GSK3B
SCHEMBL2788133 0.71 CHKA (0.51) EGFRDYRK3CLK1CLK3GSK3B
SCHEMBL4768194 0.71 BACE1 (0.36) L3MBTL1KDM4ERAB9AALDH1A1MAPT
SCHEMBL4774451 0.70 ALOX5 (0.42) L3MBTL1KDM4ERAB9AGFERALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567112-B1 THIAZOLIDIN-4-ONES FOR INHIBITING hYAK3 PROTEINS SMITHKLINE BEECHAM CORP (US) 2008-10-15 EP claimed