SCHEMBL4776074

SCHEMBL4776074

O=C1N=C(Nc2c(F)cccc2Br)SC1=Cc1cccc2cccnc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.35
RAB9A P51151 4/20 0.35
KMT2A Q03164 5/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 3/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
SLC40A1 Q9NP59 3/20 0.34
MEN1 O00255 4/20 0.33
BACE1 P56817 1/20 0.33
PPARG P37231 1/20 0.33
CISD1 Q9NZ45 1/20 0.33
KDM4E B2RXH2 3/20 0.32
AGTR1 P30556 2/20 0.32
MITF O75030 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
EGFR P00533 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2787658 0.83 DYRK3 (0.48) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL2787656 0.83 DYRK3 (0.48) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL4768194 0.80 BACE1 (0.36) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL4774451 0.76 ALOX5 (0.42) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL4765880 0.74 ROCK1 (0.43) KMT2AMEN1L3MBTL1
SCHEMBL4770530 0.73 PDE10A (0.46) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL4768062 0.72 DYRK3 (0.38) KMT2AMAPTALDH1A1GLAPOLB
SCHEMBL4772929 0.72 SLC40A1 (0.38) KMT2AMAPTPOLBSLC40A1MEN1
SCHEMBL4774422 0.71 CYP2C9 (0.36) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL2993506 0.71 CISD1 (0.39) KMT2AMAPTALDH1A1HTTSLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567112-B1 THIAZOLIDIN-4-ONES FOR INHIBITING hYAK3 PROTEINS SMITHKLINE BEECHAM CORP (US) 2008-10-15 EP claimed