SCHEMBL4766632

SCHEMBL4766632

CC(C)CC(NC(=O)OC(C)(C)C)C(=O)N(C(=O)Nc1ccccc1F)C1CCCNC[C@@H]1O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
MAPK1 P28482 1/20 0.38
AAK1 Q2M2I8 1/20 0.37
SCN9A Q15858 4/20 0.36
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PSMB5 P28074 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4762162 0.88 MAPK1 (0.41) MAPK1AAK1CTSSCTSKMEN1
SCHEMBL6593215 0.82 MAPK1 (0.36) MAPK1MEN1KMT2A
SCHEMBL6610801 0.81 MBTPS1 (0.34) NPC1
SCHEMBL6610800 0.81 MBTPS1 (0.34) NPC1
SCHEMBL6610805 0.81 CD274 (0.33) SCN9A
SCHEMBL6588445 0.81 MAPK1 (0.38) MAPK1AAK1CTSKMEN1KMT2A
SCHEMBL4212772 0.77 CTSS (0.35) MAPK1AAK1SCN9ACTSSCTSK
SCHEMBL5971691 0.76 MAPK1 (0.36) MAPK1CTSSCTSKMEN1KMT2A
SCHEMBL6611358 0.75 MAPK1 (0.36) MAPK1AAK1PSMB5
SCHEMBL4766735 0.75 CTSK (0.38) MAPK1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed