SCHEMBL6588445

SCHEMBL6588445

CC(C)CC(NC(=O)OC(C)(C)C)C(=O)N(C(=O)c1ccccn1)C1CCCNC[C@@H]1O

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
CTSK P43235 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 3/20 0.34
REN P00797 3/20 0.34
AAK1 Q2M2I8 2/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
PLA2G1B P04054 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
XBP1 P17861 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
RAB9A P51151 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5971691 0.83 MAPK1 (0.36) MAPK1CTSKSMN1; SMN2ALDH1A1REN
SCHEMBL4762162 0.83 MAPK1 (0.41) MAPK1CTSKRENAAK1MAPT
SCHEMBL4766735 0.82 CTSK (0.38) MAPK1CTSKALDH1A1REN
SCHEMBL4766632 0.81 NPC1 (0.41) MAPK1CTSKAAK1MEN1KMT2A
SCHEMBL6593215 0.79 MAPK1 (0.36) MAPK1ALDH1A1RENLMNAKDM4E
SCHEMBL6611358 0.77 MAPK1 (0.36) MAPK1ALDH1A1RENAAK1LMNA
SCHEMBL4212772 0.74 CTSS (0.35) MAPK1CTSKALDH1A1AAK1LMNA
SCHEMBL3955650 0.73 CTSL (0.36) MAPK1CTSKAAK1
SCHEMBL3955653 0.73 CTSL (0.36) MAPK1CTSKAAK1
SCHEMBL5971129 0.73 REN (0.41) MAPK1CTSKRENKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed