SCHEMBL4767404

SCHEMBL4767404

CCCc1ccccc1CSc1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
MAPT P10636 1/20 0.40
HDAC1 Q13547 1/20 0.39
TXN P10599 1/20 0.39
TXNRD1 Q16881 1/20 0.39
ADK P55263 1/20 0.38
HTR1A P08908 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
FDPS P14324 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 1/20 0.36
GRIN2B Q13224 1/20 0.36
F2RL1 P55085 3/20 0.36
NISCH Q9Y2I1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765782 0.81 HPGD (0.51) HPGDMAPTSMN1; SMN2NPC1ALDH1A1
SCHEMBL9011939 0.81 HDAC1 (0.45) HPGDADRA2AADRA2BADRA2CHDAC1
SCHEMBL9012401 0.78 HDAC1 (0.52) HPGDMAPTHDAC1FDPSSMN1; SMN2
SCHEMBL9013455 0.78 LMNA (0.41) HPGDMAPTHDAC1TXNTXNRD1
SCHEMBL9012067 0.78 HDAC1 (0.46) HPGDADRA2AADRA2BADRA2CHDAC1
SCHEMBL9012190 0.74 HDAC1 (0.44) HPGDADRA2AADRA2CHDAC1TXN
SCHEMBL229404 0.74 HDAC1 (0.53) HDAC1TAAR1NPC1ALDH1A1RAB9A
SCHEMBL9012538 0.72 HDAC1 (0.42) HPGDADRA2AADRA2CHDAC1TXN
SCHEMBL30435561 0.72 FDPS (0.41) HPGDHDAC1TXNTXNRD1TAAR1
Hydrochloric Acid SCHEMBL5155818 0.72 HDAC1 (0.52) HDAC1TAAR1SMN1; SMN2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1971596-A2 FUSED HETEROCYCLIC COMPOUNDS AND THEIR USE AS MINERALOCORTICOID RECEPTOR LIGANDS Takeda Pharmaceutical Company Limited (JP) 2008-09-24 EP disclosed
WO-2007077961-A2 FUSED HETEROCYCLIC COMPOUNDS AND THEIR USE AS MINERALOCORTICOID RECEPTOR LIGANDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-07-12 WO disclosed