SCHEMBL4767665

SCHEMBL4767665

Cc1c(C(=O)O)oc2cnccc12

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.54
KDM4E B2RXH2 5/20 0.51
ALDH1A1 P00352 2/20 0.51
GPR35 Q9HC97 1/20 0.50
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
MAPK1 P28482 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 2/20 0.45
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.42
HPGD P15428 3/20 0.42
EDNRA P25101 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
BRAF P15056 2/20 0.40
TDO2 P48775 1/20 0.40
ATM Q13315 1/20 0.40
EIF2AK3 Q9NZJ5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4985633 0.87 MCL1 (0.54) MCL1KDM4EALDH1A1GPR35LMNA
SCHEMBL15232598 0.85 LMNA (0.46) MCL1KDM4EALDH1A1LMNAHTT
SCHEMBL3603321 0.81 BRAF (0.39) KDM4EALDH1A1GPR35GAAL3MBTL1
SCHEMBL5620680 0.80 MAPT (0.44) KDM4EALDH1A1SMN1; SMN2RAB9ANPC1
SCHEMBL4859735 0.80 ALDH1A1 (0.41) KDM4EALDH1A1HTTGAAHPGD
SCHEMBL20875245 0.80 KDM5A (0.42) MCL1MAPK1BRAFTDO2EIF2AK3
SCHEMBL442779 0.75 MCL1 (0.60) MCL1KDM4EALDH1A1GPR35LMNA
SCHEMBL14793896 0.74 TDO2 (0.44) TDO2
Hydrochloric Acid SCHEMBL9789912 0.74 MCL1 (0.58) MCL1KDM4EALDH1A1GPR35LMNA
SCHEMBL14228040 0.73 IDO1 (0.64) BRAFTDO2EIF2AK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed