SCHEMBL4767685

SCHEMBL4767685

CC(C)N1CCN(CCC(=O)Nc2cc(-c3cccnc3)nc(-c3ccccn3)n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.47
ADORA2A P29274 5/20 0.47
GSK3B P49841 3/20 0.43
DYRK1A Q13627 3/20 0.43
PRCP P42785 3/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
EGFR P00533 1/20 0.42
ADORA3 P0DMS8 3/20 0.42
METAP1 P53582 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766014 0.78 ADORA1 (0.47) ADORA1ADORA2AADORA3
SCHEMBL4774987 0.76 ADORA2A (0.46) ADORA1ADORA2AGSK3BDYRK1A
SCHEMBL4773065 0.75 ADORA1 (0.43) ADORA1ADORA2ADYRK1AADORA3
SCHEMBL4773130 0.75 HDAC1 (0.45) DYRK1A
SCHEMBL4771758 0.74 ADORA1 (0.43) ADORA1ADORA2AADORA3
SCHEMBL4765953 0.74 LMNA (0.52)
SCHEMBL4769045 0.74 HDAC1 (0.48) ACHE
SCHEMBL4769061 0.73 ADORA2A (0.43) ADORA1ADORA2AADORA3
SCHEMBL4768684 0.73 ADORA2A (0.43) ADORA1ADORA2ADYRK1AEGFRADORA3
SCHEMBL3968244 0.73 MKNK1 (0.40) ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed