SCHEMBL4773183

SCHEMBL4773183

CC(C)NC(=O)N(CCCCNS(=O)(=O)c1ccc(Cl)cc1Cl)CC(NC(=O)O)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
TRPV4 Q9HBA0 6/20 0.39
CCR1 P32246 1/20 0.37
FABP4 P15090 2/20 0.36
CNR1 P21554 2/20 0.35
CNR2 P34972 2/20 0.35
PTGES O14684 1/20 0.35
PTGDR Q13258 2/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
RAB9A P51151 1/20 0.35
HPGD P15428 1/20 0.35
NLRP1 Q9C000 1/20 0.35
ITGAV P06756 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4136134 0.83 GAA (0.41) GAATRPV4CCR1FABP4CNR1
SCHEMBL4136057 0.82 GAA (0.40) GAATRPV4CCR1FABP4CNR1
SCHEMBL4136055 0.82 GAA (0.40) GAATRPV4CCR1FABP4CNR1
SCHEMBL4136813 0.82 TRPV4 (0.40) GAATRPV4CCR1PTGDRPTGDR2
SCHEMBL4134999 0.81 GSTO1 (0.44) GAATRPV4CCR1PTGDRPTGDR2
SCHEMBL4768147 0.80 CCR1 (0.42) GAATRPV4CCR1FABP4CNR1
SCHEMBL13872455 0.80 ALDH1A1 (0.41) GAATRPV4CCR1HPGD
SCHEMBL4130382 0.79 GAA (0.38) GAATRPV4CCR1FABP4CNR1
SCHEMBL4130384 0.79 GAA (0.38) GAATRPV4CCR1FABP4CNR1
SCHEMBL4136390 0.79 MAPK1 (0.40) GAATRPV4CCR1FABP4PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed