SCHEMBL4769748

SCHEMBL4769748

CCCCOC(=O)C(CN)c1ccc(O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.54
TSHR P16473 4/20 0.54
LMNA P02545 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 2/20 0.54
MAPK1 P28482 2/20 0.54
CYP2D6 P10635 1/20 0.54
NR1H2 P55055 1/20 0.54
RNASEL Q05823 1/20 0.54
ESR2 Q92731 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
MMP13 P45452 1/20 0.43
LTA4H P09960 2/20 0.42
NR5A1 Q13285 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15540843 0.87 SMN1; SMN2 (0.43) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL10353444 0.86 ESR1 (0.55) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL4448685 0.84 APP (0.48) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL11641330 0.84 ESR1 (0.49) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL8554442 0.82 ESR1 (0.48) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL10567492 0.82 LMNA (0.50) LMNASMN1; SMN2MAPK1L3MBTL1MMP9
SCHEMBL13290804 0.81 TSHR (0.57) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL388023 0.81 SMN1; SMN2 (0.60) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL10884235 0.81 LMNA (0.49) ESR1TSHRLMNASMN1; SMN2CYP1A2
SCHEMBL8554439 0.80 SMN1; SMN2 (0.49) ESR1TSHRLMNASMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1572678-A4 SUBSTITUTED N-PHENYL SULFONAMIDE BRADYKININ ANTAGONISTS ELAN PHARM INC (US) 2008-05-07 EP disclosed
EP-1572678-A2 SUBSTITUTED N-PHENYL SULFONAMIDE BRADYKININ ANTAGONISTS Elan Pharmaceuticals, Inc. (US) 2005-09-14 EP disclosed
WO-2004056319-A2 SUBSTITUTED N-PHENYL SULFONAMIDE BRADYKININ ANTAGONISTS ELAN PHARMACEUTICALS INC. (US) 2004-07-08 WO disclosed