SCHEMBL4770469

SCHEMBL4770469

O=C(O)CCCC(=O)OC(=O)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.48
SLC22A6 Q4U2R8 1/20 0.46
LMNA P02545 3/20 0.40
NFKB1 P19838 2/20 0.39
PMP22 Q01453 1/20 0.39
CAMK2A Q9UQM7 1/20 0.36
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
GABRR3 A8MPY1 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
HDAC3 O15379 1/20 0.34
GABBR2 O75899 1/20 0.34
CYP1A2 P05177 1/20 0.34
THRB P10828 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRR1 P24046 1/20 0.34
GABRB3 P28472 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28542836 0.87 LMNA (0.41) TSHRSLC22A6LMNANFKB1PMP22
SCHEMBL22605826 0.82 ALDH1A1 (0.38) TSHRALDH1A1CYP1A2KMT2A
SCHEMBL9030249 0.82 TSHR (0.60) TSHRLMNAALDH1A1KMT2A
SCHEMBL5769222 0.81 CAMK2A (0.37) TSHRCAMK2AALDH1A1GPR84FFAR1
SCHEMBL19925 0.79 SLC22A6 (0.65) TSHRSLC22A6LMNANFKB1PMP22
SCHEMBL1289888 0.79 SLC22A6 (0.65) TSHRSLC22A6LMNANFKB1PMP22
SCHEMBL4643776 0.79 ALDH1A1 (0.30) TSHRALDH1A1
SCHEMBL27501999 0.79 FAAH (0.47) LMNAALDH1A1CYP1A2KMT2A
SCHEMBL3185213 0.79 TSHR (0.40) TSHRALDH1A1KMT2A
SCHEMBL28804497 0.78 CYP2D6 (0.41) TSHRLMNANFKB1ALDH1A1GABRR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102858159-A Chemical compounds GLAXOSMITHKLINE LLC 2013-01-02 CN disclosed
EP-1648873-A4 NEUROPROTECTIVE MACROCYLIC COMPOUNDS AND METHODS FOR THEIR USE NEUREN PHARMACEUTICALS LTD (NZ) 2008-06-25 EP disclosed
EP-1648873-A2 NEUROPROTECTIVE MACROCYLIC COMPOUNDS AND METHODS FOR THEIR USE Neuronz Limited (NZ) 2006-04-26 EP disclosed
WO-2004084809-A2 NEUROPROTECTIVE MACROCYLIC COMPOUNDS AND METHODS FOR THEIR USE NEUREN PHARMACEUTICALS LTD. (NZ) 2004-10-07 WO disclosed