SCHEMBL4770638

SCHEMBL4770638

O=c1c([N+](=O)[O-])c(/C=C/c2cnn(Cc3ccccc3F)c2)n(Cc2ccncc2)c(=O)n1Cc1ccoc1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
MAPT P10636 3/20 0.32
ALDH1A1 P00352 1/20 0.32
PKM P14618 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SCD O00767 1/20 0.32
SCD5 Q86SK9 1/20 0.32
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30
PDE4A P27815 1/20 0.30
HDAC2 Q92769 1/20 0.30
HSPD1 P10809 1/20 0.30
HSPE1 P61604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770647 1.00 ADORA2A (0.33) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4766042 0.95 ALDH1A1 (0.35) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4766036 0.95 ALDH1A1 (0.35) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4762596 0.93 MAPT (0.37) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4762591 0.93 MAPT (0.37) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4763634 0.91 ADORA2A (0.35) ADORA2AADORA2BADORA1ALDH1A1SCD
SCHEMBL4763642 0.91 ADORA2A (0.35) ADORA2AADORA2BADORA1ALDH1A1SCD
SCHEMBL4794079 0.90 MAPT (0.38) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4794085 0.90 MAPT (0.38) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4767385 0.86 ADORA2B (0.38) ADORA2AADORA2BADORA1ALDH1A1SCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed