SCHEMBL4763642

SCHEMBL4763642

O=c1c([N+](=O)[O-])c(C=Cc2cnn(Cc3ccccc3C(F)(F)F)c2)n(Cc2ccncc2)c(=O)n1Cc1ccoc1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
SCD5 Q86SK9 6/20 0.34
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
TAS2R8 Q9NYW2 1/20 0.31
SCD O00767 1/20 0.30
GNRHR P30968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763634 1.00 ADORA2A (0.35) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4767385 0.96 ADORA2B (0.38) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4767375 0.96 ADORA2B (0.38) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4763420 0.93 ADORA2A (0.39) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4763418 0.93 ADORA2A (0.39) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4770647 0.91 ADORA2A (0.33) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4770638 0.91 ADORA2A (0.33) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4791802 0.90 NPBWR1 (0.40) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4791799 0.90 NPBWR1 (0.40) ADORA2AADORA2BADORA1SCD5ALDH1A1
SCHEMBL4771574 0.87 ADORA2A (0.39) ADORA2AADORA2BADORA1SCD5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed