SCHEMBL4770663

SCHEMBL4770663

CCN(CCn1c(-c2ccc(F)cc2)cc(I)c(NC(=O)C(C)NC)c1=O)Cc1ccc(F)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.35
ACKR3 P25106 1/20 0.34
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
MAOB P27338 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
TP53 P04637 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
XIAP P98170 1/20 0.31
BIRC2 Q13490 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TACR1 P25103 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
PLA2G7 Q13093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2358985 0.84 ELANE (0.35) MCHR1ACKR3ALDH1A1MAOBKDM4E
SCHEMBL2358982 0.84 ELANE (0.35) MCHR1ACKR3ALDH1A1MAOBKDM4E
SCHEMBL4774566 0.80 CES2 (0.46) ALDH1A1LMNATP53KDM4EMAPT
SCHEMBL4777094 0.77 CA12 (0.34) LMNATP53MAPTXIAPBIRC2
SCHEMBL4774551 0.76 TSPO (0.43) SMN1; SMN2CYP3A4CYP2D6PLA2G7
SCHEMBL4767533 0.71 CES2 (0.45) ALDH1A1LMNATP53KDM4EMAPT
SCHEMBL2321922 0.69 TSPO (0.47)
SCHEMBL2321927 0.69 TSPO (0.47)
SCHEMBL2358516 0.64 TACR1 (0.36) XIAPBIRC2TACR1
SCHEMBL3846281 0.62 ELANE (0.50) ALDH1A1KDM4EMAPTRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902065-A2 CYCLIC AMIDE DERIVATIVES INHIBITORS OF THE INHIBITOR OF APOPTOSIS PROTEINS, THEIR PREPARATION, AND THEIR USE Novartis AG (CH) 2008-03-26 EP claimed
WO-2006133147-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2006-12-14 WO claimed