SCHEMBL4774551

SCHEMBL4774551

CCC(NC)C(=O)Nc1c(I)cc(-c2ccc(F)cc2)n(CC(=O)N(CC)Cc2ccc(F)cc2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSPO P30536 5/20 0.43
PLA2G7 Q13093 8/20 0.34
CYP3A4 P08684 6/20 0.34
CYP2D6 P10635 6/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
MAPK14 Q16539 1/20 0.33
PDE6D O43924 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2317772 0.84 TSPO (0.46) TSPOPLA2G7PDE6D
SCHEMBL2317766 0.84 TSPO (0.46) TSPOPLA2G7PDE6D
SCHEMBL4767533 0.84 CES2 (0.45) SMN1; SMN2
SCHEMBL4770663 0.76 MCHR1 (0.35) PLA2G7CYP3A4CYP2D6SMN1; SMN2
SCHEMBL4777094 0.76 CA12 (0.34)
SCHEMBL2321927 0.75 TSPO (0.47) TSPOPDE6D
SCHEMBL2321922 0.75 TSPO (0.47) TSPOPDE6D
SCHEMBL4774566 0.73 CES2 (0.46) SMN1; SMN2
SCHEMBL2358720 0.67 ELANE (0.49)
SCHEMBL2358717 0.67 ELANE (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902065-A2 CYCLIC AMIDE DERIVATIVES INHIBITORS OF THE INHIBITOR OF APOPTOSIS PROTEINS, THEIR PREPARATION, AND THEIR USE Novartis AG (CH) 2008-03-26 EP claimed
WO-2006133147-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2006-12-14 WO claimed