SCHEMBL4771445

SCHEMBL4771445

Cc1c([N+](=O)[O-])c(=O)n(C(C)c2ccccc2)c(=O)n1CC1CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 5/20 0.45
DCTPP1 Q9H773 1/20 0.41
ALDH1A1 P00352 5/20 0.36
HPGD P15428 3/20 0.36
POLB P06746 1/20 0.35
LMNA P02545 4/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
CASP1 P29466 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
OPRM1 P35372 1/20 0.33
NPC1 O15118 1/20 0.33
MITF O75030 1/20 0.33
AGTR1 P30556 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765579 0.84 GNRHR (0.44) GNRHRDCTPP1ALDH1A1HPGDPOLB
SCHEMBL4762644 0.81 DCTPP1 (0.49) GNRHRDCTPP1ALDH1A1HPGDPOLB
SCHEMBL4762494 0.78 DCTPP1 (0.47) DCTPP1ALDH1A1HPGDPOLBLMNA
SCHEMBL4771453 0.76 ADORA3 (0.44) GNRHRALDH1A1HPGDLMNAMAPT
SCHEMBL4771274 0.76 PDE5A (0.46) GNRHRPDE5APDE4APDE4BPDE4C
SCHEMBL4769060 0.74 DCTPP1 (0.42) GNRHRDCTPP1ALDH1A1HPGDLMNA
SCHEMBL4765718 0.74 PDE4D (0.46) GNRHRPOLBLMNANPSR1KMT2A
SCHEMBL4769379 0.74 ALDH1A1 (0.42) GNRHRALDH1A1POLBLMNAMAPT
SCHEMBL4767817 0.73 PARG (0.38) GNRHRALDH1A1LMNAMAPTNPSR1
SCHEMBL4771460 0.72 PARG (0.39) GNRHRALDH1A1HPGDLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed