SCHEMBL4771624

SCHEMBL4771624

COc1ccc(C(Cc2cnc(Nc3ccc(OC)nc3)nc2Nc2ccccc2)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.46
NTRK2 Q16620 1/20 0.46
EGFR P00533 9/20 0.46
ITK Q08881 5/20 0.45
AURKA O14965 2/20 0.43
SYK P43405 2/20 0.43
MAPK9 P45984 2/20 0.42
CDK4 P11802 1/20 0.42
CDK2 P24941 1/20 0.42
MAPK10 P53779 1/20 0.42
MAPK8 P45983 1/20 0.42
NPY5R Q15761 1/20 0.42
FLT4 P35916 1/20 0.42
BTK Q06187 1/20 0.42
JAK2 O60674 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766654 0.94 CHEK1 (0.46) CHEK1NTRK2EGFRITKAURKA
SCHEMBL4774864 0.93 CHEK1 (0.50) CHEK1NTRK2EGFRITKAURKA
SCHEMBL4764815 0.86 CHEK1 (0.49) CHEK1NTRK2EGFRITKAURKA
SCHEMBL4766694 0.84 SYK (0.50) CHEK1NTRK2EGFRITKAURKA
SCHEMBL4765275 0.84 CHEK1 (0.43) CHEK1NTRK2AURKASYKMAPK9
SCHEMBL4775386 0.82 AURKA (0.49) NTRK2EGFRITKAURKASYK
SCHEMBL4770076 0.82 MAPK9 (0.45) CHEK1NTRK2MAPK9CDK4CDK2
SCHEMBL4775312 0.82 GAA (0.43) CHEK1NTRK2SYKMAPK9MAPK10
SCHEMBL4765277 0.81 SYK (0.44) CHEK1NTRK2SYKMAPK9MAPK10
SCHEMBL4772107 0.81 MAPK8 (0.57) EGFRITKAURKASYKMAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581531-B1 PYRIDINO¬2,3-D PYRIMIDINE DERIVATIVES AS SELECTIIVE KDR AND FGFR INHIBITORS HOFFMANN LA ROCHE (CH) 2008-02-27 EP claimed