SCHEMBL4772929

SCHEMBL4772929

O=C1N=C(Nc2cc(C(F)(F)F)ccc2Cl)SC1=Cc1cccc2cccnc12

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 11/20 0.38
ADRA2A P08913 1/20 0.36
NFKBIA P25963 2/20 0.36
RELA Q04206 2/20 0.36
MCL1 Q07820 2/20 0.35
MAPT P10636 3/20 0.35
TRPV1 Q8NER1 1/20 0.35
MDM2 Q00987 1/20 0.35
NPSR1 Q6W5P4 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
HSP90AA1 P07900 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ATM Q13315 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768062 0.86 DYRK3 (0.38) SLC40A1MAPTKDM4EMEN1HSP90AA1
SCHEMBL2787721 0.84 DYRK3 (0.46) ADRA2AMCL1MEN1KMT2AL3MBTL1
SCHEMBL2787724 0.84 DYRK3 (0.46) ADRA2AMCL1MEN1KMT2AL3MBTL1
SCHEMBL4774386 0.83 MEN1 (0.49) NFKBIARELAMAPTNPSR1KDM4E
SCHEMBL4768194 0.77 BACE1 (0.36) SLC40A1RELAMAPTKDM4EMEN1
SCHEMBL4770530 0.73 PDE10A (0.46) SLC40A1NFKBIARELAMAPTMDM2
SCHEMBL4772146 0.73 DYRK3 (0.54) MEN1KMT2APOLB
SCHEMBL4775509 0.73 DYRK3 (0.55) MEN1KMT2APOLB
SCHEMBL4776074 0.72 NPC1 (0.35) SLC40A1MAPTKDM4EMEN1KMT2A
SCHEMBL4775747 0.71 GPR84 (0.38) SLC40A1MEN1KMT2AL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567112-B1 THIAZOLIDIN-4-ONES FOR INHIBITING hYAK3 PROTEINS SMITHKLINE BEECHAM CORP (US) 2008-10-15 EP claimed