SCHEMBL4773571

SCHEMBL4773571

NC(C=O)C(c1ccc(Cl)cc1Cl)N1CCN(C(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 12/20 0.48
CNR2 P34972 10/20 0.48
CACNA1G O43497 1/20 0.40
CACNA2D1 P54289 3/20 0.40
CACNA1B Q00975 3/20 0.40
CACNB1 Q02641 3/20 0.40
CACNA1C Q13936 2/20 0.40
ACHE P22303 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OPRL1 P41146 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775561 0.84 MAPT (0.43) CACNA1G
SCHEMBL4773088 0.80 SIGMAR1 (0.36) CNR1CNR2CACNA2D1CACNA1BCACNB1
SCHEMBL7392463 0.77 CACNA1B (0.51) CNR1CACNA1GCACNA2D1CACNA1BCACNB1
SCHEMBL4771297 0.75 NPSR1 (0.46)
SCHEMBL4778352 0.73 ALDH1A1 (0.40) CNR1OPRM1OPRK1
SCHEMBL4774991 0.73 LMNA (0.39)
SCHEMBL4779187 0.72 MAPT (0.42)
SCHEMBL4778523 0.72 SCD (0.40) CNR1CNR2CACNA1GCACNA2D1CACNA1B
SCHEMBL4772508 0.71 CYP3A4 (0.36) CNR1CNR2CACNA1GCACNA2D1CACNA1B
SCHEMBL6167915 0.70 TP53 (0.40) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996550-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES Novartis AG (CH) 2008-12-03 EP claimed
WO-2007038459-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES NOVARTIS AG (CH) 2007-04-05 WO claimed