SCHEMBL4774577

SCHEMBL4774577

CC(C)CCc1cc(NCCc2ccccc2)nc(-c2cccc([N+](=O)[O-])c2)n1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.51
ALDH1A1 P00352 4/20 0.48
POLB P06746 3/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HRH4 Q9H3N8 1/20 0.48
ESR1 P03372 3/20 0.47
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PDE5A O76074 1/20 0.43
ABCG2 Q9UNQ0 3/20 0.43
ABCC1 P33527 1/20 0.43
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
BLM P54132 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776501 0.88 ALDH1A1 (0.51) CNR2ALDH1A1POLBMAPTMEN1
SCHEMBL4780655 0.82 ALDH1A1 (0.46) CNR2ALDH1A1POLBMAPTMEN1
SCHEMBL4775577 0.78 POLB (0.46) CNR2ALDH1A1POLBMAPTMEN1
SCHEMBL4779144 0.78 MEN1 (0.47) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL4778315 0.77 POLB (0.44) CNR2ALDH1A1POLBMAPTMEN1
SCHEMBL4778137 0.70 ALDH1A1 (0.48) CNR2ALDH1A1POLBMAPTMEN1
SCHEMBL4774224 0.70 ALDH1A1 (0.47) ALDH1A1MAPTMEN1KMT2AHRH4
SCHEMBL4774514 0.69 ALDH1A1 (0.47) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL4780661 0.69 ABCG2 (0.51) ALDH1A1POLBMAPTMEN1KMT2A
SCHEMBL13309932 0.69 HRH4 (0.60) ALDH1A1HRH4PDE5AABCG2BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed