SCHEMBL4774754

SCHEMBL4774754

Oc1cc(CCCc2ccccc2)nc(C2CCCCC2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
EPHX2 P34913 1/20 0.39
EPHX1 P07099 3/20 0.39
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP19A1 P11511 1/20 0.36
SLC18A3 Q16572 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
POLB P06746 1/20 0.36
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780410 0.84 NOS3 (0.44) PDE5ANOS3NOS1NOS2EPHX2
SCHEMBL4779107 0.81 PDE5A (0.47) PDE5ANOS3NOS1NOS2EPHX2
SCHEMBL4778365 0.81 PDE5A (0.40) PDE5ANOS3NOS1NOS2EPHX2
SCHEMBL4774100 0.79 NOS3 (0.42) PDE5ANOS3NOS1NOS2DRD2
SCHEMBL4778076 0.78 PDE5A (0.40) PDE5ANOS3NOS1NOS2DRD2
SCHEMBL14303430 0.78 PDE5A (0.40) PDE5ANOS3NOS1NOS2DRD2
SCHEMBL4778323 0.78 NOS3 (0.43) PDE5ANOS3NOS1NOS2DRD2
SCHEMBL4774683 0.76 NOS3 (0.39) PDE5ANOS3NOS1NOS2DRD2
SCHEMBL4776487 0.75 PDE5A (0.38) PDE5ANOS3NOS1NOS2EPHX2
SCHEMBL4796379 0.75 PDE5A (0.38) PDE5ANOS3NOS1NOS2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed