SCHEMBL4774100

SCHEMBL4774100

Nc1ccc(-c2cc(CCCc3ccccc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
PDE5A O76074 2/20 0.40
MAOB P27338 3/20 0.40
MEN1 O00255 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
DRD2 P14416 3/20 0.37
DRD4 P21917 3/20 0.37
DRD3 P35462 3/20 0.37
DHODH Q02127 1/20 0.36
VCP P55072 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778323 0.99 NOS3 (0.43) NOS3NOS1NOS2PDE5AMAOB
SCHEMBL4778076 0.90 PDE5A (0.40) NOS3NOS1NOS2PDE5AMEN1
SCHEMBL4778365 0.87 PDE5A (0.40) NOS3NOS1NOS2PDE5AMEN1
SCHEMBL14303430 0.87 PDE5A (0.40) NOS3NOS1NOS2PDE5AMEN1
SCHEMBL4776487 0.83 PDE5A (0.38) NOS3NOS1NOS2PDE5AALDH1A1
SCHEMBL4780443 0.83 PDE5A (0.38) NOS3NOS1NOS2PDE5AALDH1A1
SCHEMBL4796379 0.83 PDE5A (0.38) NOS3NOS1NOS2PDE5AALDH1A1
SCHEMBL4776170 0.83 CYP19A1 (0.39) NOS3NOS1NOS2PDE5AMEN1
SCHEMBL4774683 0.82 NOS3 (0.39) NOS3NOS1NOS2PDE5AMAOB
SCHEMBL4780429 0.82 MOK (0.42) MEN1ALDH1A1HPGDKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed