SCHEMBL4778076

SCHEMBL4778076

NCc1ccc(-c2cc(CCCc3ccccc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.40
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 1/20 0.39
ACP1 P24666 1/20 0.38
POLB P06746 2/20 0.37
CASP3 P42574 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
DRD2 P14416 3/20 0.36
DRD4 P21917 3/20 0.36
DRD3 P35462 3/20 0.36
HTR2A P28223 2/20 0.36
DHODH Q02127 1/20 0.35
MTOR P42345 1/20 0.35
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774100 0.90 NOS3 (0.42) PDE5ANOS3NOS1NOS2POLB
SCHEMBL14303430 0.89 PDE5A (0.40) PDE5ANOS3NOS1NOS2POLB
SCHEMBL4778365 0.89 PDE5A (0.40) PDE5ANOS3NOS1NOS2POLB
SCHEMBL4778323 0.88 NOS3 (0.43) PDE5ANOS3NOS1NOS2MEN1
SCHEMBL4776170 0.84 CYP19A1 (0.39) PDE5ANOS3NOS1NOS2MEN1
SCHEMBL4780429 0.83 MOK (0.42) MEN1ALDH1A1HPGDKMT2AADORA1
SCHEMBL4796379 0.82 PDE5A (0.38) PDE5ANOS3NOS1NOS2ALDH1A1
SCHEMBL4780443 0.82 PDE5A (0.38) PDE5ANOS3NOS1NOS2ALDH1A1
SCHEMBL4776487 0.82 PDE5A (0.38) PDE5ANOS3NOS1NOS2ALDH1A1
SCHEMBL4794991 0.81 ADRA1D (0.43) CASP3MEN1ALDH1A1KMT2AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed