SCHEMBL4774683

SCHEMBL4774683

Nc1ccc(Oc2cc(CCCc3ccccc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
MAOB P27338 3/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
PDE5A O76074 2/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
ACACB O00763 1/20 0.34
PPARG P37231 1/20 0.33
MCHR1 Q99705 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778374 0.90 NOS3 (0.38) NOS3NOS1NOS2MAOBPDE5A
SCHEMBL4774580 0.85 GRIN2B (0.40) RAB9AALDH1A1MEN1LMNAMAPT
SCHEMBL4776439 0.85 SPHK1 (0.35) PDE5AALDH1A1LMNAMAPTMCHR1
SCHEMBL4774100 0.82 NOS3 (0.42) NOS3NOS1NOS2MAOBPDE5A
SCHEMBL4778323 0.81 NOS3 (0.43) NOS3NOS1NOS2MAOBPDE5A
SCHEMBL4794914 0.80 ADRA2A (0.45)
SCHEMBL4774754 0.76 PDE5A (0.41) NOS3NOS1NOS2PDE5AKMT2A
SCHEMBL4780410 0.76 NOS3 (0.44) NOS3NOS1NOS2PDE5AKMT2A
SCHEMBL4779107 0.73 PDE5A (0.47) NOS3NOS1NOS2PDE5AALDH1A1
SCHEMBL4778076 0.73 PDE5A (0.40) NOS3NOS1NOS2PDE5AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed