SCHEMBL4775252

SCHEMBL4775252

CC(C)(C)OC(=O)NC1(C)CN(CCc2ccccc2)CC12CC2

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.47
DRD2 P14416 1/20 0.44
NPFFR1 Q9GZQ6 1/20 0.42
NPFFR2 Q9Y5X5 1/20 0.42
OPRM1 P35372 3/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
NAMPT P43490 2/20 0.39
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
AKT1 P31749 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739535 1.00 SIGMAR1 (0.47) SIGMAR1DRD2NPFFR1NPFFR2OPRM1
SCHEMBL81713 0.89 NPFFR1 (0.50) SIGMAR1NPFFR1NPFFR2CA12CA1
SCHEMBL4772739 0.78 SIGMAR1 (0.41) SIGMAR1DRD2NPFFR1NPFFR2OPRM1
SCHEMBL4772742 0.78 SIGMAR1 (0.41) SIGMAR1DRD2NPFFR1NPFFR2OPRM1
SCHEMBL27929854 0.77 NPFFR1 (0.48) SIGMAR1DRD2NPFFR1NPFFR2OPRM1
SCHEMBL27947092 0.77 NPFFR1 (0.48) SIGMAR1DRD2NPFFR1NPFFR2OPRM1
SCHEMBL5067807 0.75 DRD2 (0.45) SIGMAR1DRD2NPFFR1NPFFR2OPRM1
SCHEMBL8541686 0.75 SIGMAR1 (0.44) SIGMAR1DRD2NPFFR1NPFFR2CA12
SCHEMBL6008955 0.75 SIGMAR1 (0.44) SIGMAR1DRD2NPFFR1NPFFR2CA12
SCHEMBL739534 0.74 OPRL1 (0.37) OPRM1CTSSCTSKOPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1930321-A1 PROCESS FOR PREPARATION OF TETRASUBSTITUTED 5-AZASPIRO[2.4]- HEPTANE DERIVATIVES AND OPTICALLY ACTIVE INTERMEDIATES THEREOF Daiichi Sankyo Company, Limited (JP) 2008-06-11 EP claimed