SCHEMBL4776462

SCHEMBL4776462

CCCCCCC(CCCCCC)c1nc(CCCc2ccccc2)cc(-c2ccc(CNCCCNC(=O)OC(C)(C)C)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.40
S1PR1 P21453 5/20 0.39
S1PR3 Q99500 5/20 0.39
S1PR2 O95136 4/20 0.39
S1PR4 O95977 2/20 0.39
NPSR1 Q6W5P4 2/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
LPAR2 Q9HBW0 1/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
P2RY14 Q15391 1/20 0.37
MMP1 P03956 1/20 0.37
MMP3 P08254 1/20 0.37
MMP9 P14780 1/20 0.37
PTGES O14684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781138 0.83 S1PR1 (0.39) S1PR1S1PR3S1PR2S1PR4CNR1
SCHEMBL4795346 0.81 CTSK (0.41) CTSKNPSR1SIGMAR1BCHEP2RY14
SCHEMBL4780934 0.76 DHODH (0.40) MAPTPTGESALOX5
SCHEMBL4776475 0.76 TNKS2 (0.39) CNR1MEN1KMT2ASIGMAR1ACHE
SCHEMBL16492758 0.76 S1PR1 (0.51) CTSKS1PR1S1PR3S1PR2S1PR4
SCHEMBL6559442 0.73 ATM (0.55) CTSKNPSR1MEN1KMT2ASIGMAR1
SCHEMBL16151782 0.72 MAOA (0.56) NPSR1SIGMAR1BCHEACHE
SCHEMBL13426175 0.71 ATM (0.55) NPSR1MEN1KMT2ASIGMAR1BCHE
SCHEMBL16151781 0.69 CYP3A4 (0.46) CTSK
SCHEMBL4774621 0.69 DHODH (0.41) MAPTPTGESALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed