SCHEMBL4776571

SCHEMBL4776571

Nc1ccc(-c2nc(CCCc3ccccc3)cc(NCCc3ccccc3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.46
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
BLM P54132 1/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
PDE5A O76074 1/20 0.42
MAOB P27338 2/20 0.42
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
GBA1 P04062 1/20 0.41
HRH4 Q9H3N8 3/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774224 0.88 ALDH1A1 (0.47) ABCG2ALDH1A1MEN1KMT2AMAPT
SCHEMBL14303425 0.83 ABCG2 (0.45) ABCG2ALDH1A1MEN1KMT2AMAPT
SCHEMBL4779144 0.83 MEN1 (0.47) ABCG2ALDH1A1MEN1KMT2AMAPT
SCHEMBL14302669 0.77 BRAF (0.47) ABCG2ALDH1A1L3MBTL1BLMPDE5A
SCHEMBL13309932 0.77 HRH4 (0.60) ABCG2ALDH1A1L3MBTL1BLMPDE5A
SCHEMBL4776501 0.77 ALDH1A1 (0.51) ABCG2ALDH1A1MEN1KMT2AMAPT
SCHEMBL4778366 0.75 HRH4 (0.57) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL17407827 0.70 HRH4 (0.80) ALDH1A1HRH4HRH1
SCHEMBL11924745 0.69 MEN1 (0.58) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL4774514 0.69 ALDH1A1 (0.47) ABCG2ALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed