SCHEMBL4778366

SCHEMBL4778366

CC(C)CCc1cc(NCCc2ccccc2)nc(-c2cccc(N)c2)n1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.57
ESR1 P03372 7/20 0.51
ALDH1A1 P00352 2/20 0.45
BLM P54132 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
FYN P06241 1/20 0.42
HTR7 P34969 2/20 0.41
HRH1 P35367 1/20 0.41
RPS27 P42677 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774224 0.87 ALDH1A1 (0.47) HRH4ESR1ALDH1A1BLML3MBTL1
SCHEMBL4774760 0.83 HRH4 (0.48) HRH4ESR1ALDH1A1BLML3MBTL1
SCHEMBL4774577 0.83 CNR2 (0.51) HRH4ESR1ALDH1A1BLML3MBTL1
SCHEMBL4776571 0.75 ABCG2 (0.46) HRH4ESR1ALDH1A1BLML3MBTL1
SCHEMBL13309932 0.72 HRH4 (0.60) HRH4ALDH1A1BLML3MBTL1KDM4E
SCHEMBL14302669 0.70 BRAF (0.47) HRH4ALDH1A1BLML3MBTL1HRH1
SCHEMBL13309922 0.70 HRH4 (0.60) HRH4ALDH1A1BLML3MBTL1
SCHEMBL4776501 0.69 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL17407827 0.68 HRH4 (0.80) HRH4ALDH1A1HRH1
SCHEMBL4498447 0.67 PTGDR (0.73)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed