SCHEMBL4776930

SCHEMBL4776930

N#CCC(=O)NC(=O)Cc1ccc(N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.42
CNR2 P34972 1/20 0.42
GLS O94925 3/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CTSD P07339 1/20 0.39
MAPK8 P45983 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
CYP19A1 P11511 1/20 0.37
RORC P51449 1/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
GAA P10253 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4471126 0.83 MCL1 (0.62) MCL1CNR2ALDH1A1KDM4ECTSL
SCHEMBL15651789 0.74 CA1 (0.68) MCL1CA12CA1CA2CA9
SCHEMBL5752289 0.72 AOC2 (0.58) CNR2GLSSIGMAR1ALDH1A1CYP3A4
SCHEMBL14820608 0.72 HDAC6 (0.63) CNR2GLSSIGMAR1ALDH1A1KDM4E
SCHEMBL1632446 0.71 LMNA (0.51) CNR2GLSCTSDSIGMAR1ALDH1A1
SCHEMBL38662293 0.69 GAA (0.67) CA12CA1CA2CA9RORC
SCHEMBL18868428 0.69 ALDH1A1 (0.61) CA12CA1CA2CA9ALDH1A1
SCHEMBL9142127 0.69 MCL1 (0.62) MCL1ALDH1A1KDM4ECTSLCTSB
SCHEMBL4780769 0.69 AKR1B1 (0.50) MCL1CA12CA1CA2CA9
SCHEMBL780470 0.68 HPGD (0.49) CNR2GLSSIGMAR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008005954-A2 TRYPHOSTIN-ANALOGS FOR THE TREATMENT OF CELL PROLIFERATIVE DISEASES THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2008-01-10 WO disclosed