SCHEMBL9142127

SCHEMBL9142127

N#CCC(=O)NNC(=O)Cc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.62
ALDH1A1 P00352 5/20 0.59
KMT2A Q03164 6/20 0.56
MEN1 O00255 5/20 0.56
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
KDM4E B2RXH2 3/20 0.53
GAA P10253 2/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
EPHX2 P34913 1/20 0.50
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
POLB P06746 1/20 0.49
HTT P42858 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4471126 0.86 MCL1 (0.62) MCL1ALDH1A1KMT2AMEN1HDAC8
SCHEMBL7107935 0.84 ALDH1A1 (0.77) ALDH1A1KMT2AMEN1HDAC8HDAC6
SCHEMBL9563921 0.79 ALDH1A1 (0.75) ALDH1A1KMT2AMEN1HDAC8HDAC6
SCHEMBL19277778 0.78 MCL1 (0.69) MCL1ALDH1A1KMT2AMEN1KDM4E
SCHEMBL1529438 0.77 MCL1 (0.55) MCL1ALDH1A1KMT2AMEN1HDAC8
SCHEMBL29148895 0.77 MEN1 (0.72) ALDH1A1KMT2AMEN1HDAC8HDAC6
SCHEMBL654148 0.76 MCL1 (1.00) MCL1ALDH1A1KMT2AMEN1GAA
SCHEMBL12389341 0.76 ALOX5 (0.56) MCL1ALDH1A1KDM4EGAALMNA
SCHEMBL10612693 0.76 CTSS (0.66) MCL1ALDH1A1KMT2AMEN1HDAC8
SCHEMBL8370299 0.76 MCL1 (0.58) MCL1ALDH1A1KDM4EEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5466812-A Reacting alkyl cyanoacetate with hydrazine; catalysis, phase transfer; lactamization, cyclization BASF AKTIENGESELLSCHAFT (DE) 1995-11-14 US disclosed
EP-0413226-B1 [1,2,4]Triazo [1,5-a]pyridine BASF AG (DE) 1995-05-24 EP disclosed
EP-0628547-A1 Process for the preparation of N-aminopyridones BASF Aktiengesellschaft (DE) 1994-12-14 EP disclosed
EP-0413226-A2 [1,2,4]Triazo [1,5-a]pyridine BASF Aktiengesellschaft (DE) 1991-02-20 EP disclosed