SCHEMBL4778874

SCHEMBL4778874

Cn1c(COc2ccc3c(c2)OCCn2ncc(-c4ccncc4)c2-3)nc2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
RAB9A P51151 7/20 0.45
NPC1 O15118 6/20 0.45
PPARG P37231 3/20 0.41
PDE10A Q9Y233 4/20 0.40
PDE4B Q07343 3/20 0.39
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
PDE4A P27815 2/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780878 0.84 MAOB (0.49) SMN1; SMN2RAB9ANPC1PDE10APDE4B
SCHEMBL4780055 0.83 PDE10A (0.50) PDE10APDE4BPDE3BPDE3APDE4A
SCHEMBL4780912 0.83 PDE10A (0.47) PDE10APDE4BPDE3BPDE3APDE4A
SCHEMBL4781570 0.78 PDE10A (0.36) PDE10APDE4BPDE3BPDE3APDE4A
SCHEMBL4763295 0.76 PDE10A (0.61) RAB9ANPC1PDE10APDE4BPDE3B
SCHEMBL4781215 0.73 MAOA (0.39)
SCHEMBL30123040 0.72 RAB9A (0.56) TP53SMN1; SMN2RAB9ANPC1PDE10A
SCHEMBL4763361 0.72 RAB9A (0.56) TP53SMN1; SMN2RAB9ANPC1PDE10A
SCHEMBL30123201 0.71 PDE10A (0.60) TP53SMN1; SMN2RAB9ANPC1PDE10A
SCHEMBL5519473 0.71 PDE10A (0.60) TP53SMN1; SMN2RAB9ANPC1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4103161-B1 COMPOSITIONS AND USES THEREOF BENEVOLENTAI CAMBRIDGE LTD (GB) 2023-12-20 EP disclosed
EP-4103161-A1 COMPOSITIONS AND USES THEREOF BenevolentAI Cambridge Limited (GB) 2022-12-21 EP disclosed
CN-115484938-A Composition and use thereof 博善人工智能剑桥有限公司 2022-12-16 CN disclosed
WO-2008001182-A1 TRICYCLIC HETEROARYL COMPOUNDS AS PDE10 INHIBITORS PFIZER PRODUCTS INC. (US) 2008-01-03 WO disclosed
WO-2008001182-A1 TRICYCLIC HETEROARYL COMPOUNDS AS PDE10 INHIBITORS PFIZER PRODUCTS INC. (US) 2008-01-03 WO disclosed