SCHEMBL4730718

SCHEMBL4730718

COC(CCCn1ccnn1)c1ccc(OCc2ccc(-c3ccc(C(F)(F)F)nc3)nc2C)cc1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.34
ATP4A P20648 1/20 0.33
ATP4B P51164 1/20 0.33
ERBB2 P04626 1/20 0.33
MINK1 Q8N4C8 1/20 0.33
TRPV3 Q8NET8 12/20 0.33
GRM5 P41594 1/20 0.33
FFAR1 O14842 1/20 0.31
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4732040 0.91 TRPV3 (0.35) GRM2ATP4AATP4BERBB2MINK1
SCHEMBL4726101 0.90 TRPV3 (0.32) GRM2ATP4AATP4BERBB2MINK1
SCHEMBL4780494 0.85 ERBB2 (0.46) GRM2ATP4AATP4BERBB2MINK1
SCHEMBL4728989 0.83 TRPV3 (0.34) GRM2ATP4AATP4BTRPV3PSEN1
SCHEMBL4728771 0.83 MMP1 (0.34) GRM2ATP4AATP4BERBB2MINK1
SCHEMBL4728357 0.82 ERBB2 (0.37) GRM2ATP4AATP4BERBB2MINK1
SCHEMBL4782735 0.81 ATP4A (0.33) GRM2ATP4AATP4BERBB2MINK1
SCHEMBL4782623 0.79 PPARD (0.34) GRM2ATP4AATP4BTRPV3FFAR1
SCHEMBL4784067 0.78 PPARD (0.32) ATP4AATP4BPSEN1PSEN2APH1B
SCHEMBL4784127 0.77 PPARD (0.33) GRM2TRPV3FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO claimed
WO-2008034579-A1 2-HETEROCYCLYL-5-PHENOXYMETHYLPYRIDINE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed