SCHEMBL4782026

SCHEMBL4782026

Cc1ccccc1C(=O)c1ccnn1CCCN

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 3/20 0.40
CHRM1 P11229 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
ENPP3 O14638 1/20 0.36
ALPL P05186 1/20 0.36
XIAP P98170 1/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK1 P28482 1/20 0.35
CTNNB1 P35222 1/20 0.35
WNT3A P56704 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14160345 0.81 HTT (0.40) ALDH1A1LMNAMEN1KMT2AHTT
SCHEMBL4782961 0.77 DRD2 (0.43) MEN1KMT2AHTTCYP3A4SMN1; SMN2
SCHEMBL31646349 0.73 F2 (0.43) ELANEALDH1A1KDM4EGAAMEN1
SCHEMBL4784655 0.73 LMNA (0.45) ELANECHRM1ALDH1A1KDM4ELMNA
SCHEMBL30861065 0.69 TEAD2 (0.45) ALDH1A1KDM4ELMNAGAATSHR
SCHEMBL29387256 0.65 CYP3A4 (0.55) ALDH1A1GAAKMT2AENPP3ALPL
SCHEMBL333141 0.65 CYP3A4 (0.55) ALDH1A1GAAKMT2AENPP3ALPL
SCHEMBL19398166 0.65 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAGAACYP1A2
SCHEMBL10669335 0.63 CYP3A4 (0.59) ALDH1A1GAAKMT2AENPP3ALPL
SCHEMBL10936467 0.63 ALDH1A1 (0.47) ALDH1A1KDM4ELMNAGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed