SCHEMBL4782453

SCHEMBL4782453

Nc1cccc(-c2nc(Nc3ccc4c(cnn4C(=O)O)c3)c3ccccc3n2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 6/20 0.53
MEN1 O00255 8/20 0.52
KMT2A Q03164 8/20 0.52
RORC P51449 1/20 0.51
MAPK14 Q16539 1/20 0.51
TGFBR1 P36897 1/20 0.51
MAPT P10636 4/20 0.50
KDM4E B2RXH2 2/20 0.50
MAPK1 P28482 1/20 0.50
ABCC1 P33527 1/20 0.50
TP53 P04637 2/20 0.49
PDE5A O76074 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
SIRT5 Q9NXA8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
ROCK2 O75116 2/20 0.48
ROCK1 Q13464 1/20 0.48
KDM1A O60341 1/20 0.48
GAA P10253 1/20 0.48
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL878154 0.90 MEN1 (0.60) ABCG2MEN1KMT2ARORCMAPK14
SCHEMBL876648 0.88 ABCG2 (0.55) ABCG2MEN1KMT2ARORCMAPK14
SCHEMBL877613 0.86 ABCG2 (0.68) ABCG2MEN1KMT2AMAPTPDE5A
SCHEMBL877614 0.86 ABCG2 (0.68) ABCG2MEN1KMT2AMAPTPDE5A
SCHEMBL877856 0.86 ROCK2 (0.68) ABCG2MEN1KMT2ARORCMAPK14
SCHEMBL1724176 0.85 ROCK2 (0.52) ABCG2MEN1KMT2ARORCMAPK14
SCHEMBL1726552 0.84 ABCG2 (0.53) ABCG2MEN1KMT2ARORCMAPK14
SCHEMBL877390 0.83 MEN1 (0.50) ABCG2MEN1KMT2ARORCMAPK14
SCHEMBL877621 0.83 ROCK2 (0.45) ABCG2ABCC1ROCK2
SCHEMBL877653 0.81 ROCK2 (0.45) ABCG2ABCC1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008054599-A2 RHO KINASE INHIBITORS SURFACE LOGIX, INC. (US) 2008-05-08 WO disclosed
EP-1865958-A2 PHARMACOKINETICALLY IMPROVED COMPOUNDS Surface Logix, Inc. (US) 2007-12-19 EP disclosed
WO-2006105081-A2 PHARMACOKINETICALLY IMPROVED COMPOUNDS SURFACE LOGIX, INC. (US) 2006-10-05 WO disclosed