SCHEMBL4782663

SCHEMBL4782663

Cc1ncc(NC(=O)c2cc(C(=O)NCC3CC3)cc(C(C)(C)C)c2)cc1-n1cc(C(=O)NCC(C)(C)C)nn1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.38
EPHA3 P29320 1/20 0.38
FRK P42685 1/20 0.38
GLS O94925 7/20 0.36
KCNH2 Q12809 4/20 0.35
CACNA1I Q9P0X4 1/20 0.35
MCHR1 Q99705 3/20 0.34
DDT P30046 2/20 0.34
KIT P10721 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778561 0.85 DDT (0.45) DDT
SCHEMBL4779210 0.84 TEK (0.41) DDT
SCHEMBL4784000 0.83 DDT (0.34) DDT
SCHEMBL4780132 0.81 RAF1 (0.40)
SCHEMBL4782092 0.81 BRAF (0.34) DDTHTR1A
SCHEMBL4730805 0.81 DDT (0.42) MAPK14DDT
SCHEMBL4781066 0.79 MAPK14 (0.55) MAPK14EPHA3FRK
SCHEMBL4782901 0.79 BRAF (0.45) DDT
SCHEMBL4782957 0.78 BRAF (0.42) GLS
SCHEMBL4783784 0.78 TEK (0.40) DDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed