SCHEMBL4782092

SCHEMBL4782092

Cc1nc(-c2cc(C(=O)Nc3cnc(C)c(-n4cc(C(=O)NCC(C)(C)C)nn4)c3)cc(C(C)(C)C)c2)no1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 14/20 0.34
HTR1D P28221 3/20 0.34
SLC6A4 P31645 2/20 0.34
DDT P30046 2/20 0.33
RAF1 P04049 3/20 0.32
MEN1 O00255 2/20 0.32
MAPT P10636 2/20 0.32
KMT2A Q03164 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
HTR1A P08908 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
HTR1B P28222 1/20 0.32
HTR2A P28223 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782091 0.92 BRAF (0.32) BRAFHTR1DSLC6A4DDTMAPT
SCHEMBL4778561 0.83 DDT (0.45) DDTTP53RAB9A
SCHEMBL4779210 0.82 TEK (0.41) BRAFDDTRAF1
SCHEMBL4784000 0.82 DDT (0.34) BRAFDDTRAF1MEN1MAPT
SCHEMBL4782663 0.81 MAPK14 (0.38) DDTHTR1A
SCHEMBL14293723 0.80 MAPK14 (0.42) BRAFHTR1DSLC6A4RAF1MEN1
SCHEMBL4780132 0.79 RAF1 (0.40) BRAFRAF1
SCHEMBL4730805 0.79 DDT (0.42) BRAFDDTRAF1
SCHEMBL4783784 0.76 TEK (0.40) BRAFDDTRAF1
SCHEMBL4782901 0.75 BRAF (0.45) BRAFDDTRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed