SCHEMBL4783455

SCHEMBL4783455

COC(=O)CNC(=O)C1CN1S(=O)(=O)c1ccc(C(C)C)c(C(C)C)c1C(C)C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.36
MMP2 P08253 8/20 0.34
ADAM17 P78536 1/20 0.34
MMP1 P03956 3/20 0.33
MMP13 P45452 3/20 0.33
MMP9 P14780 2/20 0.33
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MMP3 P08254 2/20 0.32
MMP7 P09237 2/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
TRPA1 O75762 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782536 0.89 ALDH1A1 (0.36) GAAMMP2ADAM17ALDH1A1NPSR1
SCHEMBL4526832 0.78 EPHX2 (0.43) GAAMMP2ADAM17ALDH1A1
SCHEMBL4529431 0.74 MMP2 (0.56) MMP2ALDH1A1POLB
SCHEMBL13964804 0.70 HCRTR1 (0.51) GAAMAPTPOLB
SCHEMBL4530837 0.67 EPHX2 (0.44) GAAMMP2ALDH1A1NPSR1
SCHEMBL23519455 0.63 TDP1 (0.64) GAAMMP2MMP9ALDH1A1NPSR1
SCHEMBL3825925 0.62 PLAU (0.51) GAAMMP1MMP13MMP9ALDH1A1
SCHEMBL13964809 0.62 HCRTR1 (0.51) GAAMAPTTDP1POLB
SCHEMBL719443 0.61 FABP3 (0.41) ALDH1A1TRPA1
SCHEMBL9425114 0.61 SLC9A1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1985624-A2 Single step method of radiofluorination of biologically active compounds or biomolecules Bayer Schering Pharma Aktiengesellschaft (DE) 2008-10-29 EP disclosed