SCHEMBL4784918

SCHEMBL4784918

COc1ccc(C(=O)CN2C(=O)C(=O)c3cc(Br)cc(Br)c32)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARK7 Q99497 4/20 0.67
NPC1 O15118 2/20 0.58
GSK3B P49841 2/20 0.46
RAB9A P51151 2/20 0.46
PAX8 Q06710 1/20 0.46
ALDH1A1 P00352 6/20 0.44
ALDH2 P05091 4/20 0.43
ALDH3A1 P30838 4/20 0.43
CHRM5 P08912 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4783761 0.88 GSK3B (0.59) PARK7NPC1GSK3BALDH1A1ALDH2
SCHEMBL4784997 0.88 PARK7 (0.57) PARK7NPC1RAB9AALDH1A1
SCHEMBL4785634 0.84 PARK7 (0.61) PARK7NPC1GSK3BRAB9AALDH1A1
SCHEMBL4735921 0.81 PARK7 (1.00) PARK7GSK3BALDH1A1ALDH2ALDH3A1
SCHEMBL4781965 0.80 PARK7 (0.52) PARK7NPC1GSK3BRAB9AALDH1A1
SCHEMBL4786048 0.79 PARK7 (0.78) PARK7GSK3BALDH1A1ALDH2ALDH3A1
SCHEMBL4781976 0.74 PARK7 (0.71) PARK7ALDH1A1ALDH2ALDH3A1CHRM5
SCHEMBL1609155 0.74 NPC1 (1.00) NPC1GSK3BRAB9APAX8ALDH1A1
SCHEMBL9179332 0.74 ALDH1A1 (0.62) PARK7GSK3BALDH1A1ALDH2ALDH3A1
SCHEMBL18954539 0.73 ALDH1A1 (0.62) PARK7NPC1RAB9AALDH1A1ALDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074078-A1 SELECTIVELY DELIVERABLE ISATIN-BASED CYTOTOXIC AGENTS UNIVERSITY OF WOLLONGONG (AU) 2008-06-26 WO disclosed