SCHEMBL4785773

SCHEMBL4785773

Cc1nn(-c2ccccc2)nc1C(=O)N[C@H]1CCc2cccc(N3CCN(C)CC3)c2C1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.72
SCN9A Q15858 4/20 0.72
SCN5A Q14524 3/20 0.72
MTNR1A P48039 3/20 0.44
MTNR1B P49286 3/20 0.44
RIPK1 Q13546 3/20 0.41
DRD4 P21917 2/20 0.41
POLB P06746 1/20 0.41
DRD2 P14416 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
PKM P14618 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
KAT2B Q92831 1/20 0.40
MAPT P10636 1/20 0.39
TMEM97 Q5BJF2 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788501 1.00 KCNH2 (0.72) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4788123 0.86 KCNH2 (0.74) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4788313 0.84 KCNH2 (0.55) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL20288009 0.84 SCN9A (1.00) KCNH2SCN9ASCN5APOLBDRD2
SCHEMBL7027930 0.81 MTNR1A (0.65) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL7027929 0.81 MTNR1A (0.65) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL841303 0.81 SCN9A (0.71) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL840155 0.81 SCN9A (0.57) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4789252 0.80 KCNH2 (0.50) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4788131 0.79 TRPV4 (0.49) KCNH2SCN9ASCN5AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO claimed
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed