SCHEMBL4785787

SCHEMBL4785787

Clc1cccc(Nc2ccsc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FADS1 O60427 6/20 0.45
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP1B1 Q16678 1/20 0.43
KMT2A Q03164 5/20 0.43
MAPT P10636 4/20 0.43
MEN1 O00255 4/20 0.43
ALDH1A1 P00352 3/20 0.43
GAA P10253 3/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
KDM1A O60341 1/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
ROCK1 Q13464 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1686631 0.82 FADS1 (0.59) FADS1KMT2AMAPTMEN1ALDH1A1
SCHEMBL27877680 0.78 CNR1 (0.43) CYP1A1CYP1A2CYP1B1KMT2AMAPT
SCHEMBL28066532 0.78 CYP3A4 (0.60) CYP1A2KMT2AMAPTMEN1ALDH1A1
SCHEMBL3185782 0.77 CYP2A6 (0.36) ALDH1A1TDP1GRIK1
SCHEMBL30342506 0.76 MEN1 (0.68) FADS1CYP1A2KMT2AMAPTMEN1
SCHEMBL3951892 0.76 MEN1 (0.68) FADS1CYP1A2KMT2AMAPTMEN1
SCHEMBL3038796 0.76 HSD17B10 (0.57) CYP1A2KMT2AMAPTMEN1ALDH1A1
SCHEMBL27668399 0.75 TDP2 (0.62) KMT2AMAPTMEN1ALDH1A1LMNA
SCHEMBL30080248 0.74 MEN1 (0.54) CYP1A1CYP1A2CYP1B1KMT2AMAPT
SCHEMBL11349013 0.73 ADRA2A (0.38) KMT2AMAPTMEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008089307-A2 DELTA 5 DESATURASE INHIBITORS FOR THE TREATMENT OF PAIN, INFLAMMATION AND CANCER LEXICON PHARMACEUTICALS, INC. (US) 2008-07-24 WO disclosed
WO-2008089310-A2 DELTA 5 DESATURASE INHIBITORS FOR THE TREATMENT OF OBESITY LEXICON PHARMACEUTICALS, INC. (US) 2008-07-24 WO disclosed