SCHEMBL4786035

SCHEMBL4786035

NCOc1ccn(C(=O)O)n1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTT P42858 1/20 0.33
SCN4A P35499 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21438893 0.79 HTT (0.32) ALDH1A1NPSR1HTTSMN1; SMN2
SCHEMBL21439236 0.79 PKM (0.33) ALDH1A1NPSR1HTTSMN1; SMN2
SCHEMBL21245097 0.78 NUDT1 (0.38) HTTSMN1; SMN2
SCHEMBL21438556 0.77 HTT (0.31) HTTSMN1; SMN2
SCHEMBL21244926 0.76 MEN1 (0.33) HTTSMN1; SMN2
SCHEMBL21438906 0.76 SIGMAR1 (0.31) HTT
SCHEMBL26667193 0.76 EPHX2 (0.41)
SCHEMBL21438610 0.74 L3MBTL1 (0.31)
SCHEMBL22392306 0.73 CFTR (0.39)
SCHEMBL20239860 0.73 L3MBTL1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008132502-A1 PYRAZOLYL-AMINO-SUBSTITUTED PYRIMIDINES AND THEIR USE FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-11-06 WO disclosed
WO-2008117050-A1 PYRAZOLYL-AMINO-SUBSTITUTED PYRAZINES AND THEIR USE FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-10-02 WO disclosed