SCHEMBL4786167

SCHEMBL4786167

CC(O)(c1ccc(F)cc1)c1ccc(CN(C(=O)c2cccnc2)c2ccc(F)cc2)cn1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
TSHR P16473 1/20 0.51
PTGDR2 Q9Y5Y4 1/20 0.46
MLYCD O95822 1/20 0.44
POLB P06746 1/20 0.44
HTT P42858 1/20 0.44
MAPK14 Q16539 2/20 0.42
CXCR2 P25025 1/20 0.42
PDK1 Q15118 5/20 0.40
NR1H4 Q96RI1 1/20 0.39
CYP3A4 P08684 1/20 0.39
PTGES O14684 1/20 0.39
ALOX5 P09917 1/20 0.39
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
RORC P51449 1/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4738966 0.91 GAA (0.54) GAATSHRPTGDR2MLYCDPOLB
SCHEMBL4735056 0.88 GAA (0.50) GAATSHRPTGDR2MLYCDPOLB
SCHEMBL4737668 0.87 GAA (0.56) GAATSHRPTGDR2MLYCDPOLB
SCHEMBL4737592 0.81 GAA (0.56) GAATSHRPTGDR2POLBHTT
SCHEMBL4737107 0.81 GAA (0.58) GAATSHRPTGDR2POLBHTT
SCHEMBL4737949 0.78 GAA (0.52) GAATSHRPTGDR2MLYCDPOLB
SCHEMBL4738200 0.77 GAA (0.51) GAATSHRPTGDR2MLYCDPOLB
SCHEMBL4737583 0.77 GAA (0.46) GAATSHRPTGDR2POLBHTT
SCHEMBL4739768 0.76 GAA (0.55) GAATSHRMLYCDHTTPDK1
SCHEMBL4738239 0.76 TSHR (0.49) GAATSHRPTGDR2POLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed