SCHEMBL4786331

SCHEMBL4786331

CC(C)c1nc(NS(=O)(=O)c2ccccc2)cc2c1C(=O)OCC2

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 0.42
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GAA P10253 4/20 0.38
TSHR P16473 2/20 0.38
MAPT P10636 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CXCR2 P25025 1/20 0.37
MAPK1 P28482 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PIK3CD O00329 1/20 0.35
HTT P42858 1/20 0.35
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786337 0.91 PKM (0.43) PKMKDM4EALDH1A1HPGDGAA
SCHEMBL4788073 0.90 HSD11B1 (0.41) PKMKDM4EALDH1A1TSHRMAPT
SCHEMBL4787522 0.90 PKM (0.44) PKMKDM4EALDH1A1GAAMAPT
SCHEMBL4787350 0.74 KDM4E (0.45) PKMKDM4EALDH1A1
SCHEMBL4788782 0.74 KDM4E (0.46) PKMKDM4ETSHRLMNASMN1; SMN2
SCHEMBL4747016 0.72 MAOA (0.34)
SCHEMBL18238925 0.66 MAOA (0.36)
SCHEMBL25352139 0.62 GAA (0.58) PKMKDM4EALDH1A1HPGDHSD17B10
SCHEMBL1381858 0.62 PDE4A (0.73) PKMKDM4EALDH1A1HPGDHSD17B10
SCHEMBL4069470 0.61 MAOA (0.37) KDM4EGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed