SCHEMBL4787522

SCHEMBL4787522

CC(C)c1nc(NS(=O)(=O)c2ccc(Cl)cc2)cc2c1C(=O)OCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 0.44
MAPT P10636 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
HSD11B1 P28845 1/20 0.41
DRD2 P14416 2/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
DRD3 P35462 2/20 0.39
HTR6 P50406 2/20 0.39
KDM4E B2RXH2 4/20 0.39
LMNA P02545 3/20 0.39
CXCR2 P25025 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786337 0.91 PKM (0.43) PKMMAPTL3MBTL1HSD11B1KDM4E
SCHEMBL4786331 0.90 PKM (0.42) PKMMAPTHSD11B1KDM4ELMNA
SCHEMBL4788073 0.90 HSD11B1 (0.41) PKMMAPTHSD11B1KDM4ELMNA
SCHEMBL4747016 0.74 MAOA (0.34)
SCHEMBL4788782 0.74 KDM4E (0.46) PKML3MBTL1HSD11B1KDM4ELMNA
SCHEMBL4787350 0.70 KDM4E (0.45) PKML3MBTL1KDM4EALDH1A1KMT2A
SCHEMBL4749246 0.69 DYRK1A (0.36) GAA
SCHEMBL4063663 0.64 MAOA (0.31)
SCHEMBL4786333 0.64 CA1 (0.33)
SCHEMBL18238925 0.64 MAOA (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed