SCHEMBL4786447

SCHEMBL4786447

COC(=O)[C@H](Cc1ccc(-n2cc(C)c3cccnc32)cc1)NC(=O)c1c(Cl)cncc1Cl

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 12/20 0.49
PDE4A P27815 3/20 0.46
KCNH2 Q12809 2/20 0.46
ITGB1 P05556 11/20 0.43
ITGB7 P26010 4/20 0.42
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
ITGA5 P08648 1/20 0.41
CNR2 P34972 2/20 0.39
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CNR1 P21554 1/20 0.37
ITGA2 P17301 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733110 0.91 ITGA4 (0.59) ITGA4PDE4AKCNH2ITGB1ITGB7
SCHEMBL12889776 0.78 ITGA4 (0.48) ITGA4ITGB1ITGB7ITGA2
SCHEMBL7428016 0.74 ITGA4 (0.58) ITGA4ITGB1ITGB7ITGB3ITGAV
Hydrochloric Acid SCHEMBL6510331 0.73 ITGA4 (0.57) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4786565 0.73 ITGA4 (0.58) ITGA4ITGB1
SCHEMBL4730881 0.72 ITGA4 (0.53) ITGA4ITGB1ITGB7
SCHEMBL13819259 0.69 ITGA4 (0.54) ITGA4ITGB1ITGB7
SCHEMBL4783431 0.69 ITGA4 (0.59) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4734982 0.69 ITGA4 (0.49) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL4735439 0.69 ITGA4 (0.65) ITGA4ITGB1ITGB7ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed