SCHEMBL7428016

SCHEMBL7428016

COC(=O)[C@H](Cc1ccc(N)cc1)NC(=O)c1c(Cl)cncc1Cl

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.58
ITGB1 P05556 16/20 0.58
ITGB7 P26010 4/20 0.51
LNPEP Q9UIQ6 1/20 0.48
ITGB3 P05106 1/20 0.47
ITGAV P06756 1/20 0.47
ITGA5 P08648 1/20 0.47
ATM Q13315 1/20 0.43
TYMS P04818 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6510331 0.99 ITGA4 (0.57) ITGA4ITGB1ITGB7LNPEPITGB3
SCHEMBL295783 0.88 ITGB1 (0.53) ITGA4ITGB1ITGB7LNPEPITGA5
SCHEMBL1240417 0.88 ITGB1 (0.53) ITGA4ITGB1ITGB7LNPEPITGA5
Hydrochloric Acid SCHEMBL7391192 0.87 ITGB1 (0.52) ITGA4ITGB1ITGB7LNPEPITGA5
SCHEMBL7428248 0.86 ITGA4 (0.76) ITGA4ITGB1ITGB7ITGB3ITGAV
SCHEMBL7424019 0.82 LNPEP (0.41) ITGA4ITGB1LNPEPATM
SCHEMBL27542813 0.81 ITGB1 (0.60) ITGA4ITGB1ITGB7LNPEP
SCHEMBL6639882 0.81 ITGB1 (0.60) ITGA4ITGB1ITGB7LNPEP
SCHEMBL6515360 0.81 ITGB1 (0.67) ITGA4ITGB1
SCHEMBL28742827 0.80 ITGB1 (0.46) ITGA4ITGB1ITGB7LNPEPITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020035127-A1 Phenylalanine derivatives CELLTECH THERAPEUTIS, LIMITED 2002-03-21 US disclosed
US-6329372-B1 HETEROCYCLIC AMIDE COMPOUNDS ARE ABLE TO INHIBIT THE BINDING OF ALPHA4 INTEGRINS TO THEIR LIGANDS AND ARE OF USE IN THE PROPHYLAXIS AND TREATMENT OF IMMUNE OR INFLAMMATORY DISORDERS. CELLTECH THERAPEUTICS LIMITED (GB) 2001-12-11 US disclosed
EP-1051399-A1 PHENYLALANINE DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTS CELLTECH THERAPEUTICS LIMITED (GB) 2000-11-15 EP disclosed
WO-1999037618-A1 PHENYLALANINE DERIVATIVES USEFUL AS PHARMACEUTICAL AGENTS CELLTECH THERAPEUTICS LIMITED (GB) 1999-07-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020035127-A1 Phenylalanine derivatives PAH, VCAM1, IL4I1 ITGA4 5/4885ITGB1 8/4885ITGB7 25/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.