SCHEMBL4734982

SCHEMBL4734982

CCOC(=O)[C@H](Cc1ccc(Nc2ncccc2N)cc1)NC(=O)c1c(Cl)cncc1Cl

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 18/20 0.49
ITGB1 P05556 18/20 0.49
ITGB3 P05106 1/20 0.42
ITGAV P06756 1/20 0.42
ITGA5 P08648 1/20 0.42
CYP3A4 P08684 1/20 0.41
ITGB7 P26010 2/20 0.41
ITGA2 P17301 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4735069 0.91 ITGB1 (0.41) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL4735360 0.86 ITGA4 (0.62) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL4733396 0.80 KLK5 (0.41) ITGB1ITGB3ITGAV
SCHEMBL4736051 0.78 ITGB1 (0.54) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL7428016 0.76 ITGA4 (0.58) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL5366913 0.75 ITGB1 (0.54) ITGA4ITGB1
Hydrochloric Acid SCHEMBL6510331 0.75 ITGA4 (0.57) ITGA4ITGB1ITGB3ITGAVITGA5
SCHEMBL4736663 0.74 ITGB1 (0.44) ITGA4ITGB1CYP3A4
SCHEMBL7538523 0.74 ITGB1 (0.59) ITGA4ITGB1ITGA5ITGB7ITGA2
SCHEMBL4786565 0.73 ITGA4 (0.58) ITGA4ITGB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO claimed
WO-2008064823-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-06-05 WO disclosed