SCHEMBL4786822

SCHEMBL4786822

O=C(O)C1CCCN(c2nc(-c3cccc(O)c3)nc(N3CCc4ccccc4C3CO)n2)C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
IDH2 P48735 1/20 0.39
PIK3CA P42336 9/20 0.39
PIK3CD O00329 2/20 0.37
PIK3CB P42338 2/20 0.37
PIK3CG P48736 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
POLB P06746 1/20 0.37
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
TSHR P16473 2/20 0.36
AKR1C3 P42330 1/20 0.35
AKR1C1 Q04828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782541 0.91 DGAT2 (0.40) HSD17B10ALDH1A1LMNAMAPTMAPK1
SCHEMBL4784742 0.88 PIK3CA (0.42) HSD17B10ALDH1A1PIK3CAPIK3CDPIK3CB
SCHEMBL4785055 0.87 PIK3CA (0.39) IDH2PIK3CAPIK3CBESR1ESR2
SCHEMBL4785045 0.87 PIK3CA (0.39) IDH2PIK3CAPIK3CBESR1ESR2
SCHEMBL4782397 0.84 PIK3CA (0.39) IDH2PIK3CAESR1ESR2
SCHEMBL4782618 0.84 PIK3CA (0.40) PIK3CAPIK3CDPIK3CBPIK3CGESR1
SCHEMBL4782625 0.84 PIK3CA (0.40) PIK3CAPIK3CDPIK3CBPIK3CGESR1
SCHEMBL4786826 0.82 KDM4E (0.43) HSD17B10KDM4EALDH1A1MEN1KMT2A
SCHEMBL4784691 0.82 AOC3 (0.41) PIK3CAESR1ESR2
SCHEMBL4783343 0.82 AOC3 (0.41) PIK3CAESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed