SCHEMBL4787156

SCHEMBL4787156

O=C1CSC(C2=COC(Cc3ccccc3)O2)N1c1ccc(Oc2ccc(Cl)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GFER P55789 2/20 0.43
KCNA5 P22460 1/20 0.41
MAPT P10636 1/20 0.41
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KMT2A Q03164 3/20 0.39
METAP1 P53582 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743532 0.77 GFER (0.70) ALDH1A1HTTNPSR1GFERCA1
SCHEMBL747924 0.76 KMT2A (0.53) ALDH1A1HTTNPSR1MAPTKMT2A
SCHEMBL4743542 0.74 ALDH1A1 (0.52) ALDH1A1HTTNPSR1GFERKCNA5
SCHEMBL748256 0.74 HCRTR1 (0.55) ALDH1A1KMT2AMEN1
SCHEMBL4743949 0.72 ALDH1A1 (0.64) ALDH1A1HTTNPSR1GFERMAPT
SCHEMBL4745876 0.71 CA1 (0.61) ALDH1A1HTTNPSR1GFERMAPT
SCHEMBL4746811 0.71 MAPT (0.59) ALDH1A1HTTNPSR1GFERMAPT
SCHEMBL4746660 0.71 ALDH1A1 (0.59) ALDH1A1HTTNPSR1GFERMAPT
SCHEMBL4743525 0.70 CA1 (0.56) ALDH1A1HTTNPSR1GFERMAPT
SCHEMBL4747930 0.70 MAPT (0.55) ALDH1A1HTTNPSR1GFERMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO claimed
WO-2008112674-A1 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-09-18 WO disclosed